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Ele investigheaza un evantai bogat de cunostinfe, adre- siindu-se difertelor componente ale procesului cognitiv, Asemenea teste asigura o notare rapid, permitind evaluarea unui numar mare de studenti sau medici, in conditile unui ) solubilitatea in apa ©) coeficientul de-partaj fipidelapa, ) pKa mic; ©) afinitat portor pentru un sistem trans- 2. Care dintre urmitoarele afirmatii pri- vind ecuatia Henderson-Hasselbach 4) indiedproportia absorbyiei_ prin filtrare pentru moleculele hidro- solubile; b) indic& proportia legarii- medic Imentelor de proteinele plasmatice; lied proportia de ionizare toase administeata al ©) permite caleularea timp d ‘mate a uneisubstanye medic iecare intrebare din cele de mai jos contine 5 raspunsuri posibile 3. Care dintre urmatoarele afirma Privind legarea medicamentelor de proteinele plasmatice nu este coreeta 4) legarea se face numai de globw line; ») legarea este un proces reversibil (dinamic); ©) legarea prin covalente reprezinta situafii de except; 4) medicamentele slab active, prin competitc, se pot deplasa de pe proteine ©) medicamentele legate de prote- inele plasmatice nu pot traversa ‘membranele prin fltrare a) substanta. medic forma de solutie apoasa, in eazul tramuset medicamentoas’i sub forma de suspensie apoasa, in D.Oiee ©) monitorizarea medicamentelor in- {roduse in terapeuticd, Indeosebi a reactilor adverse; 4) studiul terapeutie intensiv in etapa 4) evaluarea parametrilor farmacoci netici pentru medicamentele noi; b) stabilitea indiceluiterapeutic; alll-aa evaluat clinice; ) precizarea interactiunilor medica- rmentoase. intrebari de tip complement grupat Instruetiuni: Piecare intrebare din cele de mai jos contine 5 sugesti de raspuns dintre ite pot i corecte 2 sau 3, Raspundetifolosind urmatoarea cheie A, dacia, b, © sunt corecte; BB, dacd a d, sunt eorecte , daca by, d, sunt corecte: , daca a, e sunt corecte ©) tranzitimestinal lent U1. Care dintre urmatoarele afirmati defines biodisponibilita 23. Care dintre urmatoarele caracte- ristici ale preparatelor farmaceu- tice pot favoriza absorbi a) exprima fractiunea din doza ad- ste hidrosolubilt; ») exprima tract ‘ministrata care ajunge in singe; ©) exprima fractiunea din doza admi- nistrat care se dizolv la locul ab- sorbjii «t) exprima proportia din doza admi- histraaldlsponibi pentru actiune; fractiunea din doza ad- ‘ministrat care este fipasolubila, 4) structura macromolecular’; b) proportia mare a forme neioni- zate in cazul electrolifilor; ©) structura peptidica in cazul admi- nistei orale; <) pKa mare in cal acizilor organi ©) pKa mare in cazul bazelor orzanice 24. Care dintre urmitoarele afirmatit sunt corecte pentru filtrare (trece- rea prin canalele membranare) ca tuna din modalittile de traversare a membranelor: factori pot itatea dupa ad- 1) modificiri patologice ale mucoasei digestive, a) are foc numai penteu moteculele +) Legare in proportie mare de prote ‘miei hidrosotubile incle plasmatice b) se face un consum de enery var in intestin sau ha pi ° mul pasaj hepatic ansportor specializat Formacologie generala 26, Difuziunea medicamentelor prin re este depen= 8) gradul de jonizare mic; ') pKa-ul substan ©) pul medina 4) prezenta unui sistem transportor specializat; 20, Traversarea membranelor celulare prin transport specializat: 1) are loc ta nivelul canalelor mem- branare; bb) se face eu consum de energie; ©) este posibilé numa pentru mole- calle hidrosolubile; 14) poate fi influentata prin competi- tie moleeulara; ©) are loc numai in sensul gradien- tului de concentratie sau de po- tential electrochimie. (et nat 1) absorbtie rapi permite absorbs temic ionizate; ie posibila administrarea de sub- fe ritante; istrarea sublingual are ur- ele avantaje: moleculelor pu 1) este conditionata de hidrosolubi- Titate; ©) evitt inaetivarea la primul pasa} hepatic. 2. ul aparent de distributie al bstanfe: medicamentoase se lculeaza findnd seama de: 2) ritmal epurari ) doza administrata ©) eradul de acurmutare in anumite tesutur 4d) concentraia plasmatie; ©) peoportialegaii de albuminele plasmatice u 29. Epurarea prin metabolizare se face ups o cinetic# de ordinul I In doze miei si dupa o cineticd de ordinul 0 la doze mari in cazul me- dicamentelor: a) salicilatis ») fenitoina; ©) dicumarotu 4) digoxina;, ) etanolul; 30. Se elimina prin bili sub forma ac- tiv in cantitati semnificative: 1) ampicilina ') penicilina G; 6) tetraciclinele; 4) eritromici ©) gentamicina, 34. Potential foarte mare de a provoca dependent psihied au ) amfetamina; ») nicotina; ) morfina: 4) cocaina; e) cafeina; 32. Au tendinta mare de a dezvolta to leranta si dependenta fiziea: 8) morfina: ») cocaina: ©) nicotina; 4) amfetamina; ©) alcoolul etc. agB2- Se pot obfine efete de tip retard (aepozit prin: 4) implantarea subeutanata de pelete; b) administrarea rectal de supozi- toare ©) injectarea intramuscular’ de solu- tituleioase: 4) injectarea intramusculard de sus- P €) administrarea prin inkalajie de ae rosoli i microctis 34, Care dintre urmatoarele afirms dicamentelor dupi 0 cinetic de ‘ordinul I: a) constanta de epurare (proprie ‘medicamentului) se exprima prin 0,693 «1/2 b) timpul de obfinere a concentra tiei constante (In platou) depinde de doza administratt; ©) marirea geometries a dozei deter- mind o crestere aritmetica a dura tei concentratiei eficace; 4) epurarea este practic terminata dupa o perioada de 4 ori mai mare decattimpal la Tajunnatstire; ©) durata mentinerii unei concentra cficace terapeutic de medicament relatia: Ke 36. 4) hemoliza produsa de nitrofurani; b) tulburarile auditive si vestibulare produse de antibioticele aminogli- cozidice; ©) socul anafilactic produs de pent cine; 44) agranulocitoza produsa de amino- fenazona;, ) apneea la doze mici de suxame- toniu, Care dintre urmatoarele afirmatii sunt coreete pentru reaetille ad- verse de tip ei 4) apar datorits unor particularitti de comportare farmacocinetic’ by sunt independente de dora; ©) sunt careacteristi telor cu 0 toxicitateintrinseca mare i un indice trap medicamen- 37. 38. Farmacologie. Te autoovaluare 4) sunt inercigate pentru compusit Inrudit structural; ©) prezenfa lor este mare in conditile administariimedicamentelor pe cale oral, fn tratamental reactitor alergice medicamentoase in functie de sit aie se utilizeaz a) antihistaminice b) adrenalin’ ©) glucocorticoizi; ) antinflamatori nesteroidiene; ©) atropina, Care dintre urmatorii factor pot favoriza aparitia reactiilor adverse de tip toxie: 4) indice terapeutic mic; ») defictul organelor de epurare; ©) interactiunimedicamentoase cu fect sinergic: 4) contactul preslabil cu substanta activa, ©) volum de distibutie mare. Pentru histamina sunt corecte ur mitoarele afiematii: a) se elibereaza in urma reactied an- tigen/anticorp:; ») este o eatecholamina biogens; ©) intervine in controll stimulator al secrefie gastrice acide; 4) stimuleazt musculatura neteda bronsiea: ©) se gaseste in concentra mari in plachete. Awstrweti Faimacologie generals Intrebari de tip asociere compus& Alegeti pentru fiecare noyiune notata cu litere de la a) la e), enunturile Jovivitenotate cu I 512. Raspundeti conform urmatoarei scheme: A, daca se potriveste 1, daca se pouriveste 2 , dc se potrivese ambele (1 $i 2). 1 daca nu se potriveste nici I nici 2 40. |. poate produce reactii adverse idi- > produce frecvent reactii adverse alergice, 4) suecinolina; }) benzilpenicitina; ©) sulfametoxidiazina; 1) acidul acetilsalicitie; «) tetracietina AA. 1 poate produce agramulocitoza ) are © bund biodisponibilitate dupa ‘administrare oral (peste 50%), 1) cloramfenicolul (baz), ) tubocurarina; ©) elonidina; 4) metitiouracil; ©) fenilbutazona. 42. 1. se read oral 2, se administreaza iv. 4) diazepamul; b) nitrogticerina; «) succinileotin: «) oxidul de magnes ©) metoxifluranul 43. 1, se administreaza iv 2. se administreaza im. 8) benzilpenicil 45. 4) beclometazona dipropion: «) neomicina, . 1. poate deplasa de pe protenele plas- ‘matice alte medicamente 2. modified actvitatea enzimelor mi: crozomiale hepatice 2) rifampicina; b) fenilbutazona; ©) digoxina; 4) acenocumarolul; «) fenobarbitall 1. poate provoca retenfie hidrosalins 2. poate produce uleeratii ale mu consei gastric. .) carbenoxolona; ) fenilbutazona; ) lidoeaina; 4) hidrocortizonul; ©) dexametazona, este inactivata in tubul di ceste metabolizaté In masurd: mare la primal pasa) hepatic a) indometacina, by benzilpenicilit ©) lidocaina, «) oxitocina ©) izoprenalina mn Farmacologie. Teste de autoevaluare Faimacologie general Is 4___ Farmacologie. Teste de autoevaluare_ 47.1. deficitul de pompa cardiaed con- ©) acid aceilslicitie + anticoagulan- ick medicamentul te orale: bronsic contraindiea medi- 4) tolbutamida + propranotol; ceamentul ©) codeina + dionina intrebari de tip asociatie simpla 2) tubocurarina; ty pene 81. 1. nu patrunde intracelular fy eeeere 2, este metabolizata de etre colines- Instrwetiuni: Alezeti pent fecare din nofumile nota cu cife de I la 5, enuatul 3 eri teraze. ‘1 Mai potrivit din cele notate cu litere de la a la e. ) verapamil: «) atropina, pai : i 2 posts Hy rans 9) ering. fines din doa ine : 2, transport specatizat; prin intermediul siste~ Willi ipomodulinetor. Enzima intervine in procesul de formare a eicosanoidelor si PAM ilu, swiacoide eu proprietatiproinflamatori RASPUNSURI 4. Raspuns corect: b. Traversarea membranelor celulare prin filtrare presupune trece= am ‘ea moleculelor prin porit sau eanalele apoase si este conditioantd de hidrosolubi titatea medicamentelor side dimensiunea mica (Mr sub 200 micron). ‘coreet: ¢. Rifampicina induce biosinteza enzimelor microzomiale hepatice ‘Heinbolizante ale unor medicamente, carora le favorizesza metabolizarea, fenomen fae poate teractiuni medicamentoase 2. Rasy Réspuns corect: . Ecuatin Hendesson-Hasselbach permite calcularea. propor Won ice, epetv onze, m lector, pe basa pala diferite valori ale pH-ului, * " = om ccoreet: ¢, Antidotul in caz de supradozare cu heparind este sulfatul de hind, © polipeptida bazica care neutralizeaz® specific gruprile acide ale mole- Wiel le heparina, responsabite de efectul anticoagulant 3. Rilspuns corect: a. Substanjele medicamentoase se leaga in singe in special de albumine; fractiunite globulinice fixeaza rar medicamente, ele leaga specific uncle substante endoge ns corect: d. Cimetiina,biocantthistaminergic, nhiba enzimele metabo- ile le anor medicament, erescnd riscultoxie al acestore. In eazulasocieri Wetec teoiina, de exemple, tcoftinemia crest, ceen ce impune uneori Fiera soe de bronhodiatator ‘4. Raspuns coreet: b. O substanta ca si se poatd absorbi trebuie si se gascasca sub forma dizolvata ta locul absorbtiei. in cazul suspensiilor apoase injectate intra Wisp ‘muscular dizolvarea este lenta, aceste substanfe realizand forme farmaceutice de Aepozit (retard. ‘coreet: b. Guanetidina (neurosimpatolitic) patrunde in terminatile simpa- © le paralizeaza) folosind mecanismul ce asigura recaptarea noradrenal W© quanctiina gi simpatomimeticele indirecte - efedrind, amfetamind - exist un ‘Aviaqonism competitiv pentru mecanismultransportor prin membrana, 5. Raspuns corect: . in cazulinjectriintravenoase nu se pune problema absorbieh substanfa medicamentoast este introdusa direct in circulate, WAspuns coreet:c. Furosemidul administat in doze mari potenjeaz8 efectul toni- 6. . f Ailineckor asupra automatismalui etopie. Consecutv creste riscularitmilor, cauza Raspums corect: c, Noradrenalin (norepinefrna) prin oxidare (sub actiunea MAO) Ail ipokatiemia generat de diureza excesiva e transforma in normetanefrind, un metabolit inactiv fermacodinamic. Wispuns corcet: d. Propranololul scade marcat fuxul sanghin fa nivelul ficatului consecutiv clearence-ul hepatic al tidocainei, creseindu-i concentratia ‘phiatich 51 crescand riscul apartie de reaciitoxice. 7. Raspuns corect: c. Marea majortate a medicamentelor se epureaz dupa o cinetich de ordinul 1 (cinetics exponential), proporjia epurat& find intotdeauna fix in atea de timp, pentru @ anumita substanta . Recomandarile OMS la care fara noastra a aderat previd moni- 8. Raspuns corect: e. Medicamentele polare find insolubile in tipide, nu tree prin uiiyarea medicamentefor dupa introducerea in terapeutic3 insistind asupea deceit rembrane gi deci nu se absorb practic in cazul administririt orale. Controlul sence a reactilor adverse, mentratiei lor in plasma nu are sens corect: C(b, d). Biodisponibiltatea exprima proportia din cantitatea de administratt disponibila pentru actiune si practic reprezinta fractiunea istrata care ajunge in sing 8. Raspuns corect: b. Manitolul acjioncazs\ ca diuretic prin mecanism osmotic, dech specific dn doz ads HE Waspuns corect: Bla, c, d). Biodisponibilitatea poate fi micgorata prin leziunile ‘iesises intestinal care interfer absorb, prin inactvarea nor medicaments de hive ack cloridec i enzimele digestive, sau prin bioinativarea la priml pass Heputc, Forma tarmaceuict necorespunzitoare poate fio alti cau de Woiaponiitate vedas 10. Rispuns coreet: a Modificarea fluidititii membranelor neuronale, produsa de exemplar de eat cele locale, este un fenon ‘de macromolecule receptoare. ‘corect: ¢. 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