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Opioid Analgesics
Receptor Stimulation Mu
P hysical dependence E uphoria A nalgesia R espiratory depression kappa S edation A nalgesia (spinal) M iosis delta Analgesia
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DEPRESSION :
1- Respiratory centre depression Both rate and depth of respiration are diminished Dangerous in Head injury and asthmatics 2- cough center depressed 3- Vasomotor centre high doses cause fall in BP and .1 bradycardia